199853-75-3

Upstream product

• 24424-99-5 di-tert-butyl dicarbonate 

Downstream Products

• 168957-42-4 (R)-6-amino-1-methyl-4-(3-methylbenzyl)hexahydro-1,4-diazepine 
• 199853-77-5 {[(R)-3-[tert-Butoxycarbonyl-(3-methyl-benzyl)-amino]-2-(toluene-4-sulfonylamino)-propyl]-methyl-amino}-acetic acid ethyl ester 
• 199853-78-6 {Methyl-[(S)-3-(3-methyl-benzylamino)-2-(toluene-4-sulfonylamino)-propyl]-amino}-acetic acid ethyl ester 
• 199853-74-2 4-Methyl-N-[(R)-1-methyl-4-(3-methyl-benzyl)-[1,4]diazepan-6-yl]-benzenesulfonamide 
• 1026269-55-5 (3-Methyl-benzyl)-[(S)-1-(toluene-4-sulfonyl)-aziridin-2-ylmethyl]-carbamic acid tert-butyl ester 

Relevant academic research and scientific papers

Asymmetric synthesis of (R)-6-amino-1-methyl-4-(3-methyl- benzyl)hexahydro-1H-1,4-diazepine from L-asparagine

An efficient asymmetric synthesis of (R)-6-amino-1-methyl-4-(3- methylbenzyl)hexahydro-1H-1,4-diazepine [(R)-2] which serves as the amine part of (R)-1, a potent and selective 5-HT3 receptor antagonist, is described. Formation of the hexahydro-