200949-84-4Relevant academic research and scientific papers
Synthesis of gastrin antagonists, analogues of the C-terminal tetrapeptide of gastrin, by introduction of a β-homo residue
Rodriguez,Fulcrand,Laur,Aumelas,Bali,Martinez
, p. 522 - 528 (2007/10/02)
A series of analogues of Boc-Trp-Leu-Asp-Phe-NH2, a potent gastrin agonist, were synthesized by introducing a β-homo residue in the sequence. These compounds were tested in vivo on acid secretion, in the anesthetized rat, and for their ability
