20242-40-4Relevant articles and documents
Synthesis and antibacterial activity of novel 5-(heteroaryl)isoxazole derivatives
RamaRao, R. Janaki,Rao, A.K.S. Bhujanga,Sreenivas,Kumar, B. Suneel,Murthy
, p. 243 - 250 (2011/06/26)
The synthesis, characterization and antibacterial activity of novel isoxazole derivatives were reported. 3-Di (alkylamino)acryloalkanones were prepared and used as synthons to get the target isoxazole derivatives via reaction with hydroxylamine hydrochloride or hydroxylamine-O-sulphonic acid.
A Regioselective Synthesis of 3,5-Disubstituted Isoxazoles
Yokoyama, Masataka,Tsuji, Kouichi,Kushida, Mari
, p. 67 - 72 (2007/10/02)
The 3-aryl-5-, and 5-aryl-3-(phenylsulphonylmethyl)isoxazoles (6) and(9) respectively were regioselectively prepared from 1-aryl-3-methylthio-4-phenylsulphonylbut-2-en-1-one (1).As an application of the present method, 3-methyl-5-(4-.pyridyl)isoxazole (2)