211761-80-7Relevant articles and documents
1,3-Disubstituted benzazepines as novel, potent, selective neuropeptide Y Y1 receptor antagonists
Murakami, Yasushi,Hara, Hirokazu,Okada, Tetsuo,Hashizume, Hiroshi,Kii, Makoto,Ishihara, Yasunobu,Ishikawa, Michio,Shimamura, Mayumi,Mihara, Shin-Inchi,Kato, Goro,Hanasaki, Kohji,Hagishita, Sanji,Fujimoto, Masafumi
, p. 2621 - 2632 (2007/10/03)
A novel series of potent and selective non-peptide neuropeptide Y (NPY) Y1 receptor antagonists, having benzazepine nuclei, have been designed, synthesized, and evaluated for activity. Chemical modification of the R1 and R3 substitue