215121-76-9Relevant academic research and scientific papers
Design, synthesis, and structure-activity relationships of substituted piperazinone-based transition state factor Xa inhibitors
Su, Ting,Yang, Hua,Volkots, Deborah,Woolfrey, John,Dam, Suiko,Wong, Paul,Sinha, Uma,Scarborough, Robert M.,Zhu, Bing-Yan
, p. 729 - 732 (2007/10/03)
The structure-activity relationship of a novel series of substituted piperazinone-based factor Xa inhibitors is described. The most potent compound 34 displays IC50 of 0.9 nM.
