217489-00-4

Upstream product

• 2338-71-8 5-fluoro-1H-indole-3-carbaldehyde 
• 98-59-9 p-toluenesulfonyl chloride 

Downstream Products

• 217489-03-7 trans-β-<5-fluoro-1-(p-tolylsulfonyl)indol-3-yl>acrylic acid 
• 468717-78-4 trans-3-[5-fluoro-1-(4-toluenesulfonyl)-1H-indol-3-yl]-N-methoxy-N-methylacrylamide 
• 1383575-19-6 (5-fluoro-1-tosyl-1H-indol-3-yl)methanol 
• 1383575-47-0 C₃₅H₄₁FN₆O₅S 
• 1383575-20-9 3-Bromomethyl-5-fluoro-1-(toluene-4-sulfonyl)-1H-indole 

Relevant academic research and scientific papers

Synthesis and serotonin receptor affinities of a series of trans-2- (indol-3-yl)cyclopropylamine derivatives

A series of four racemic ring-substituted trans-2-(indol-3- yl)cyclopropylamine derivatives was synthesized and tested for affinity at the 5-HT(1A) receptor, by competition with [3H]-8-OH-DPAT in rat hippocampal homogenates, and for affinity at

Gold(I)-catalyzed dearomative rautenstrauch rearrangement: Enantioselective access to cyclopenta[ b ]indoles

A highly enantioselective dearomative Rautenstrauch rearrangement catalyzed by cationic (S)-DTBM-Segphosgold(I) is reported. This reaction provides a straightforward method to prepare enantioenriched cyclopenta[b]indoles. These studies show vast differenc

Di/tri-aza-spiro-C9-C11alkanes

The invention relates to compounds of the formula I [in-line-formulae]A-D-C(R1)2—B??(I),[/in-line-formulae] in which the substituents are as defined in the specification; in free form or in salt form; to its preparation, to its use as medicament and to medicaments comprising it.

DI/TRI-AZA-SPIRO-C9-C11ALKANES

The invention relates to compounds of the formula I A-D-C(R1)2-B (I), in which A and B are aromatic ring systems and wherein D is selected from the groups D1 to D5 and the other substituents are as defined in the specification; in free form or in salt form; to its preparation, to its use as medicament and to medicaments comprising it.