218297-75-7Relevant academic research and scientific papers
Design of a high affinity peptidomimetic opioid agonist from peptide pharmacophore models
Wang, Chenguang,McFadyen, Iain J.,Traynor, John R.,Mosberg, Henry I.
, p. 2685 - 2688 (2007/10/03)
A pair of diastereomeric peptidomimetics based upon opioid receptor- binding pharmacophore models derived for a series of opioid tetrapeptide was synthesized. Both analogues display high opioid receptor affinity, moderate selectivity for the μ opioid rece
