220285-03-0

Basic information

• Product Name: [(1R,3S)-3-(6-amino-9H-purin-9-yl)cyclopentyl]methanol
• Synonyms: cyclopentanemethanol, 3-(6-amino-9H-purin-9-yl)-, (1R,3S)-
• CAS NO: 220285-03-0
• Molecular Formula: C₁₁H₁₅N₅O
• Molecular Weight: 233.2697
• Mol File: 220285-03-0.mol
• Article Data: 5

Chemical Properties

• Boiling Point: 505.2°C at 760 mmHg
• Flash Point: 259.3°C
• Density: 1.62g/cm³
• Vapor Pressure: 4.99E-11mmHg at 25°C
• Refractive Index: 1.804
• CAS DataBase Reference: [(1R,3S)-3-(6-amino-9H-purin-9-yl)cyclopentyl]methanol(CAS DataBase Reference)
• NIST Chemistry Reference: [(1R,3S)-3-(6-amino-9H-purin-9-yl)cyclopentyl]methanol(220285-03-0)
• EPA Substance Registry System: [(1R,3S)-3-(6-amino-9H-purin-9-yl)cyclopentyl]methanol(220285-03-0)

Safety Data

• Hazardous Substances Data: 220285-03-0(Hazardous Substances Data)

Upstream product

• 158799-92-9 (1R,cis)-4-(6-amino-9H-purin-9-yl)-2-cyclopentene-1-methanol 
• 168960-19-8 (1S,4R)-1-amino-4-hydroxymethyl-2-cyclopentene hydrochloride 
• 200002-41-1 (-)-[(1R,4S)-tert-butyl 3-oxo-2-azabicyclo(2.2.1)hept-5-ene-2-carboxylate] 
• 153011-43-9 (1S,cis)-tert-butyl N-[4-(hydroxymethyl)-2-cyclopenten-1-yl]carbamate 
• 158799-91-8 (1R,cis)-4-(6-chloro-9H-purin-9-yl)-2-cyclopentene-1-methanol 
• 287473-95-4 (1R,cis)-4-[(5-Amino-6-chloro-4-pyrimidinyl)amino]-2-cyclopentene-1-methanol 
• 130931-83-8 (1S,4R)-2-azabicyclo[2,2,1]hept-5-en-3-one 
• 87-42-3 6-chloropurine 
• 192118-38-0 (1R,2R,3S,4S)-4-(tert-butoxymethyl)-2,3-(isopropylidenedioxy)cyclopentan-1-ol 
• 212911-15-4 (1S,4R)-4-(tert-butoxymethyl)-1-hydroxycyclopent-2-ene 
• 212911-13-2 (1S,4R)-1-benzyloxy-4-(tert-butoxymethyl)cyclopent-2-ene 
• 212911-11-0 (1R,2R,3S,4S)-1-benzyloxy-2,3-dihydroxy-4-(tert-butoxymethyl)cyclopentane 
• 212911-19-8 (1'S,4'S)-9-[4-(tert-butoxymethyl)cyclopent-2-enyl]adenine 
• 212911-17-6 (1'S,4'R)-9-[4-(tert-butoxymethyl)cyclopent-2-enyl]-6-chloropurine 

Relevant articles and documents

Synthesis of D- And L-carbocyclic nucleosides via rhodium-catalyzed asymmetric hydroacylation as the key step

(Chemical Equation Presented) D- and L-carbocyclic nucleosides were obtained by a new procedure involving an enantioselective rhodium/duphos- catalyzed hydroacylation reaction as the key step. The 3-hydroxymethyl- cyclopentanol intermediate was obtained by stereoselective reduction of ketone and by dynamic kinetic resolution (DKR).

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