220932-72-9Relevant academic research and scientific papers
Modulations of the amide function of the preferential dopamine D3 agonist (R,R)-S32504: Improvements of affinity and selectivity for D3 versus D2 receptors
Peglion, Jean-Louis,Poitevin, Christophe,La Cour, Clotilde Mannoury,Dupuis, Delphine,Millan, Mark J.
body text, p. 2133 - 2138 (2009/12/25)
Starting with the preferential dopamine (DA) D3 agonist S32504, we prepared two series of derivatives of the general formula I-A and I-B, in an effort to improve both potency and selectivity. For the first set of derivatives, where the primary
Disubstituted trans-3,4,4a,5,6,10b-hexahydro-2H-naphth[1,2-b]-1,4-oxazines
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, (2008/06/13)
New compounds of formula: wherein: A represents alkyl, alkenyl, alkynyl, cycloalkylalkyl or aralkyl, and E represents: in racemic form or in the form of optical isomers, and the addition salts thereof with pharmaceutically acceptable acids. Those compounds may be used as medicaments.
