233608-04-3Relevant articles and documents
N-(diethoxyphosphoryl)aldimines as synthetic equivalents of A1 type synthons
Zwierzak, Andrzej,Napieraj, Anna
, p. 93 - 96 (2007/10/03)
Novel organophosphorus reagents useful for convergent synthesis of primary amines are presented.
Synthesis of α-arylalkylamines by addition of Grignard reagents to N- (diethoxyphosphoryl)aldimines
Zwierzak, Andrzej,Napieraj, Anna
, p. 930 - 934 (2007/10/03)
Addition of organomagnesium bromides to N-(diethoxyphosphoryl) aldimines 1 carded out in tetrahydrofuran at 20-25°C affords diethyl N-alkyl- phosphoramidates 2a-w in high yields and spectroscopic purity. Deprotection of the latent amino groups in 2 results in the formation of α-arylalkylamine hydrochlorides 3a-w.