2341740-84-7Relevant articles and documents
Highly Selective PTK2 Proteolysis Targeting Chimeras to Probe Focal Adhesion Kinase Scaffolding Functions
Popow, Johannes,Arnhof, Heribert,Bader, Gerd,Berger, Helmut,Ciulli, Alessio,Covini, David,Dank, Christian,Gmaschitz, Teresa,Greb, Peter,Karolyi-?zguer, Jale,Koegl, Manfred,McConnell, Darryl B.,Pearson, Mark,Rieger, Maria,Rinnenthal, Joerg,Roessler, Vanessa,Schrenk, Andreas,Spina, Markus,Steurer, Steffen,Trainor, Nicole,Traxler, Elisabeth,Wieshofer, Corinna,Zoephel, Andreas,Ettmayer, Peter
, p. 2508 - 2520 (2019)
Focal adhesion tyrosine kinase (PTK2) is often overexpressed in human hepatocellular carcinoma (HCC), and several reports have linked PTK2 depletion and/or pharmacological inhibition to reduced tumorigenicity. However, the clinical relevance of targeting