243844-53-3Relevant academic research and scientific papers
A convenient and versatile route to hydroquinolines by inter- and intramolecular Aza-Diels-Alder pathways
Steinhagen, Henning,Corey
, p. 1928 - 1931 (2007/10/03)
Surprisingly, the simplest method possible for o-azaxylylene production, base-induced elimination of hydrogen chloride from amide or sulfonamide derivatives of o-(chloromethyl)aniline, has never been reported. This powerful approach provides easy and stereoselective access to polycyclic hydroquinolines, as shown for an example in Equation (1).
