246177-41-3Relevant academic research and scientific papers
Peptidyl aldehyde inhibitors of calpain incorporating P2-proline mimetics
Donkor, Isaac O.,Korukonda, Rajani,Huang, Tien L.,LeCour Jr., Louis
, p. 783 - 784 (2003)
Four new peptidyl aldehydes bearing proline mimetics at the P2-position were synthesized and studied as inhibitors of calpain I, cathepsin B, and selected serine proteases. The ring size of the P2-constraining residue influenced the
