247130-39-8Relevant academic research and scientific papers
A general method for deprotection of N-toluenesulfonyl aziridines using sodium naphthalenide
Bergmeier, Stephen C.,Seth, Punit P.
, p. 6181 - 6184 (2007/10/03)
Deprotection of a variety of N-tosylaziridines with sodium naphthalenide provided the corresponding N-H-aziridines in excellent yield. No single electron transfer (SET) induced aziridine ring opening was seen under the conditions employed for the deprotection reaction.
Synthesis of optically pure 2-Aziridinemethanols: Versatile synthetic building blocks
Fujii,Nakai,Habashita,Hotta,Tamamura,Otaka,Ibuka
, p. 2241 - 2250 (2007/10/02)
Synthesis of three cis-trans pairs of N-sulfonylated-2-aziridinemethanols starting from (S)-threonine, (R)-allothreonine, a chiral 2-amino alcohol, or enantiomerically enriched 2,3-epoxy alcohols is described. A synthetic route to N-tosyl- and N-mesyl-2-a
