25462-37-7Relevant academic research and scientific papers
Enantiopure hydroxymethylated cycloalkenols as privileged small molecular multifunctional scaffolds for the asymmetric synthesis of carbocycles
Kumar, Rajan,Rej, Rohan Kalyan,Halder, Joydev,Mandal, Haridas,Nanda, Samik
, p. 498 - 512 (2016)
Enantiopure hydroxymethylated cycloalkenols bearing a quaternary stereocenter have been synthesized by a Pybox mediated enantioselective desymmetrization method. The synthesized cycloalkenols serve as starting precursors for the construction of several ch
Internally Masked Neopentyl Sulfonyl Ester Cyclization Release Prodrugs of Acamprosate, Compositions Thereof, and Methods of Use
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Page/Page column 40, (2009/04/24)
Internally masked neopentyl sulfonyl ester prodrugs of acamprosate, pharmaceutical compositions comprising such prodrugs, and methods of using such prodrugs and compositions thereof for treating diseases are disclosed. In particular, acamprosate prodrugs
Total synthesis of (+/-)-acetomycin and design of esterase-resistant analogs.
Uenishi,Kobayashi,Komine,Okadai,Yonemitsu,Sasaki,Yamada
, p. 517 - 523 (2007/10/03)
The synthesis of acetomycin and related analogs was investigated. Acetomycin was synthesized from diethyl allyl(methyl)malonate in 6.5% yield over 18 steps. The total number of steps was improved compared to our previous synthesis; i.e., four steps shorte
