261-90-5Relevant academic research and scientific papers
AZAPHENOTHIAZINES AND AZAPHENOXAZINES AS ANTIOXIDANTS
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Paragraph 00125, (2018/10/24)
The present disclosure relates generally to antioxidants. More particularly, the present disclosure relates to lubricating compositions comprising an antioxidant.
Synthesis and antitubercular activity of phenothiazines with reduced binding to dopamine and serotonin receptors
Madrid, Peter B.,Polgar, Willma E.,Toll, Lawrence,Tanga, Mary J.
, p. 3014 - 3017 (2008/02/07)
Analogs of the psychotropic phenothiazines were synthesized and examined as antitubercular agents against Mycobacterium tuberculosis H37Rv. The compounds were subsequently counter-screened for binding to the dopaminergic-receptor subtypes D1, D2, D3 and the serotonergic-receptor subtypes 5-HT1A, 5-HT2A, and 5-HT2C. The most active compounds showed MICs from 2 to 4 μg/mL and had overall reduced binding to the dopamine and serotonin receptors compared to chlorpromazine and trifluoperazine.
