2827-95-4Relevant academic research and scientific papers
One-pot synthesis of N-fused 1,2,4-triazoles and related heterocycles via I2/TBHP-mediated oxidative C–N bond formation
Wu, Yachuang,Yang, Yifeng,Qi, Yinliang,Du, Shimei,Zhang, Yongsheng,Ding, Liang,Zhao, Yanfang
supporting information, p. 4216 - 4220 (2018/10/26)
A metal-free iodine/TBHP-mediated oxidative C–N bond formation for the one-pot synthesis of N-fused 1,2,4-triazoles and related heterocycles via cyclization has been developed. This reaction which is amenable to scale-up affords the corresponding products with good to excellent yields and tolerates a wide range of functional groups.
Cu-catalysed direct C-H (hetero)arylation of [1,2,4]triazolo[4,3-a]pyridine to construct deep-blue-emitting luminophores
Wu, Jie,You, Qiulin,Lan, Jingbo,Guo, Qiang,Li, Xiaoyu,Xue, Ying,You, Jingsong
supporting information, p. 5372 - 5375 (2015/05/20)
Cu-catalysed direct C-H (hetero)arylation of [1,2,4]triazolo[4,3-a]pyridine has been accomplished for the first time to streamline the synthesis of 3-aryl-[1,2,4]triazolo[4,3-a]pyridines for screening blue-emitting materials. On this basis, the photophysi
An environmentally benign and solvent-free synthesis of 3-aryl[1,2,4]triazolo[4,3-a]pyridines and 1-aryl-5-methyl[1,2,4]triazolo[4,3-a] quinolines using phenyliodine bis(trifluoroacetate) or iodobenzene diacetate
Kumar
experimental part, p. 1237 - 1243 (2012/08/08)
A simple, solvent-free and effective method for oxidative cyclization of 2-pyridyl- and 2-quinolylhydrazones with phenyliodine bis(trifluoroacetate) and iodobenzene diacetate to the corresponding 3-aryl[1,2,4]triazolo[4,3-a]pyridines and 1-aryl[1,2,4]tria
Palladium-catalyzed coupling of aldehyde-derived hydrazones: Practical synthesis of triazolopyridines and related heterocycles
Thiel, Oliver R.,Achmatowicz, Michal M.,Reichelt, Andreas,Larsen, Robert D.
supporting information; experimental part, p. 8395 - 8398 (2010/12/25)
The palladium-catalyzed intermolecular coupling of aldehyde-derived hydrazones with chloroazines, followed by oxidative cyclization under mild conditions afforded access to a broad variety of bicyclic heterocyclic scaffolds (see scheme) that have potentia
Palladium-catalyzed chemoselective monoarylation of hydrazides for the synthesis of [1,2,4]Triazolo[4,3-a]pyridines
Reichelt, Andreas,Falsey, James R.,Rzasa, Robert M.,Thiel, Oliver R.,Achmatowicz, Michal M.,Larsen, Robert D.,Zhang, Dawei
supporting information; experimental part, p. 792 - 795 (2010/04/06)
(Chemical Equation Presented) An efficient and convenient method for the synthesis of [1,2,4]triazolo[4,3-a]pyridines was exemplified by the synthesis of 20 analogues bearing a variety of substituents at the 3-position. The methodology involves a palladiu
