2875-27-6Relevant academic research and scientific papers
Convenient synthesis of flavanone derivatives via oxa-Michael addition using catalytic amount of aqueous cesium fluoride
Miura, Motofumi,Shigematsu, Karin,Toriyama, Masaharu,Motohashi, Shigeyasu
supporting information, (2021/10/25)
A total of 36 flavanones, which included polycyclic aromatic and heterocyclic rings, were readily synthesized via oxa-Michael addition from the corresponding hydroxychalcones with a catalytic amount of aqueous cesium fluoride solution under mild conditions. This method could be applied to the scalable synthesis of eriodictyol as a known potent inhibitor of the SARS-CoV-2 spike protein.
Photochemical behavior of 2'-hydroxychalcone derivatives having pyridyl and quinolyl groups
Aizawa, Fumiya,Shinozaki, Yukino,Ishida, Yuka,Arai, Tatsuo
, p. 572 - 579 (2017/04/10)
2'-Hydroxy chalcone derivatives having heteroaromatic rings have been synthesized and their photochemical and photophysical properties have been examined in terms of tautomer produced by intramolecular hydrogen atom transfer reaction.
Inhibitory Kinetics of Azachalcones and their Oximes on Mushroom Tyrosinase: A Facile Solid-state Synthesis
Radhakrishnan, Sini K.,Shimmon, Ronald G.,Conn, Costa,Baker, Anthony T.
, p. 531 - 538 (2016/06/01)
A solid-state-based mechanochemical process was used to synthesize novel azachalcones and their oximes as tyrosinase inhibitors. Their inhibitory activities on mushroom tyrosinase using l-3,4-dihydroxyphenylalanine as a substrate were investigated. Two of
