299949-01-2Relevant articles and documents
Synthesis of [3H]-labelled 4-[ethyl[2,5,6-trimethyl-7-(2,4,6- trimethylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2,3-[3H]-butan-1- ol: A high affinity radioligand for the corticotropin-releasing hormone type 1 receptor
Hiebel, Anne-Cecile,Partilla, John S.,Rothman, Richard B.,Jacobson, Arthur E.,Rice, Kenner C.
, p. 635 - 640 (2007/10/03)
[3H]-Labelled 4-[ethyl[2,5,6-trimethyl-7-(2,4,6-trimethylphenyl) pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2,3-[3H]-butan-1-ol (3b) was prepared as a novel non-peptidic radiolabelled high affinity antagonist of the corticotropin-releasing
Synthesis of [3H](4-fluorobutyl)propyl[2,5,6-trimethyl-7-(2,4,6-trimethylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]amine: A potent radioligand for corticotropin-releasing hormone type 1 receptor
Hsin, Ling-Wei,Webster, Elizabeth L.,Chrousos, George P.,Gold, Philip W.,Eckelman, William C.,Contoreggi, Carlo,Rice, Kenner C.
, p. 899 - 908 (2007/10/03)
[3H](4-Fluorobutyl)propyl[2,5,6-trimethyl-7-(2,4,6-trimethylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]amine ([3H]LWH-154), a novel potent radiolabelled analog of the nonpeptide corticotropin-releasing hormone type 1 receptor (CRHR1/s