300698-10-6Relevant academic research and scientific papers
Visible-light-promoted C[sbnd]N and C[sbnd]S bonds formation: A catalyst and solvent-free photochemical approach for the synthesis of 1,3-thiazolidin-4-ones
Ali, Shabir,Ansari, Khursheed,Ansari, Mohd Danish,Nazeef, Mohd,Shivhare, Km Neha,Siddiqui, I. R.,Tiwari, Saurabh K.,Yadav, Vikas
, (2020/01/02)
A visible-light-induced, one-pot mild and efficient, multicomponent-tandem synthesis of diversified 1,3-thiazolidin-4-ones under catalyst and solvent-free conditions is reported. Here, visible-light, an ideal source of energy, has been used as photochemic
Tromethamine organocatalyzed efficient tandem-multicomponent synthesis of new thiazolyl-4-thiazolidinones in aqueous medium
Bhosle, Manisha R.,Kharote, Sayali A.,Bondle, Giribala M.,Mali, Jyotirling R.
supporting information, p. 1286 - 1300 (2019/04/30)
The catalytic potential of tris(hydroxymethyl)aminomethane (Tromethamine) has been assessed for the one pot three component tandem reaction involving a thiazolylmethoxy phenyl/aromatic carboxaldehyde, substituted amines and thioglycolic acid to form new t
Facile synthesis of 1,3-thiazolidin-4-ones as antitubercular agents
Subhedar, Dnyaneshwar D.,Shaikh, Mubarak H.,Arkile, Manisha A.,Yeware, Amar,Sarkar, Dhiman,Shingate, Bapurao B.
supporting information, p. 1704 - 1708 (2016/07/27)
We have developed, highly efficient, one-pot, solvent-free, [Et3NH][HSO4] catalyzed multicomponent reaction protocol for the synthesis of 1,3-thiazolidin-4-ones in excellent yields. For the first time, the 1,3-thiazolidin-4-ones were evaluated in vitro for their antimycobacterial activity against Mycobacterium tuberculosis dormant MTB H37Ra and Mycobacterium bovis BCG strains. Among the synthesized basic 1,3-thiazolidin-4-ones, particularly the compounds 4c, 4d, 4e, 4f, 4h, 4i and 4j displays promising antitubercular activity along with no significant cytotoxicity against the cell lines MCF-7, A549 and HCT-116.
Synthesis of 1,3-thiazolidin-4-one using ionic liquid immobilized onto Fe3O4/SiO2/Salen/Mn
Sadeghzadeh, Seyed Mohsen,Malekzadeh, Maryam
, p. 46 - 51 (2015/02/05)
An efficient and general method has been developed for synthesis of 1,3-thiazolidin-4-ones using magnetite nanoparticles immobilized Salen-Mn-ionic liquids as an efficient and recyclable catalyst. The inorganic, magnetic, solid base catalyst was characterized via N2 sorption, TEM, VSM, TGA, XRD, FTIR, and UV-vis. Nanocatalyst can be easily recovered by a magnetic field and reused for subsequent reactions for at least 6 times with less deterioration in catalytic activity.
Nano-Fe3O4@SiO2 supported ionic liquid as an efficient catalyst for the synthesis of 1,3-thiazolidin-4-ones under solvent-free conditions
Azgomi, Naghmeh,Mokhtary, Masoud
, p. 58 - 64 (2015/02/05)
A magnetically supported ionic liquid on Fe3O4@SiO2 nanoparticles (MNPs@ SiO2-IL) was synthesized and evaluated as a recoverable catalyst for the one-pot synthesis of 1,3-thiazolidin-4-ones in high to excellent yield under solvent-free conditions. The MNPs@SiO2-IL catalyst was characterized via Fourier transform infrared spectroscopy (FT-IR), X-ray diffraction (XRD), thermal gravimetric analysis (TGA), transmission electron microscopy (TEM) and vibrating sample magnetometer (VSM). Moreover, the catalyst could be easily recovered by magnetic separation and recycled for 10 times without significant loss of its catalytic activity.
One-pot rapid synthesis of thiazole-substituted pyrazolyl-4-thiazolidinones mediated by diisopropylethylammonium acetate
Khillare, Lalit D.,Bhosle, Manisha R.,Deshmukh, Amarsinh R.,Mane, Ramrao A.
, p. 8955 - 8964 (2015/02/19)
A convenient one-pot, rapid and scalable synthetic protocol has been developed for recently reported anti-inflammatory agents, thiazole-substituted pyrazolyl-4-thiazolidinones. Quantitative multicomponent cyclocondensation of 3-(4-methyl-2-substituted thi
Ionic liquid mediated and promoted eco-friendly preparation of thiazolidinone and pyrimidine nucleoside-thiazolidinone hybrids and their antiparasitic activities
Zhang, Xinying,Li, Xiaoyan,Li, Dongfang,Qu, Guirong,Wang, Jianji,Loiseau, Philippe M.,Fan, Xuesen
scheme or table, p. 6280 - 6283 (2010/08/06)
Without any catalyst, 2,3-disubstituted-1,3-thiazolidin-4-one derivatives were synthesized efficiently via the three-component reaction of aldehyde, amine and mercaptoacetic acid in [bmim][PF6]. The whole procedure is simple and straightforward
Kinetics of formation of 4-thiazolidinones by cyclocondensation reaction of Schiff bases and thioglycolic acid
Lawande,Arbad
, p. 352 - 354 (2007/10/03)
Kinetics of formation of 4-thiazolidinone by cyclocondensation of Schiff bases (SB) and thioglycolic acid (TGA) have been studied. The reaction shows first order dependence both on SB and TGA concentrations; it follows an overall second order kinetics. Th
