312914-89-9Relevant academic research and scientific papers
N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1)
Jetter, Michele C.,McNally, James J.,Youngman, Mark A.,McDonnell, Mark E.,Dubin, Adrienne E.,Nasser, Nadia,Zhang, Sui-Po,Codd, Ellen E.,Colburn, Ray W.,Stone, Dennis R.,Brandt, Michael R.,Flores, Christopher M.,Dax, Scott L.
, p. 2730 - 2734 (2008)
High throughput screening of our compound library revealed a series of N-pyridyl-3-benzamides as low micromolar agonists of the human TRPV1 receptor. Synthesis of analogs in this series led to the discovery of a series of N-quinolin-3-yl-benzamides as low
