3392-30-1Relevant academic research and scientific papers
Synthesis and biological activity of N-terminal lipidated and/or fluorescently labeled conjugates of astressin as corticotropin releasing factor antagonists
Rijkers, Dirk T.S.,Den Hartog, Jack A.J.,Liskamp, Rob M.J.
, p. 5099 - 5106 (2007/10/03)
This report describes the synthesis of eight N-terminally modified astressin analogs and their biochemical evaluation as corticotropin releasing factor (CRF) antagonists. The lipidated astressin derivatives were tested on rat CRF receptor type 1 and 2α an
