343615-76-9

Upstream product

• 95-23-8 5-amino-1,3-dihydro-benzoimidazol-2-one 
• 343616-21-7 1-chlorosulfonyl-piperidine-2S-carboxylic acid 4-phenyl-butyl ester 

Relevant academic research and scientific papers

An efficient synthesis of sulfamides

Here we report an efficient synthesis of sulfamides. 3,5-Lutidine was found to be an optimal solvent and catalyst for the reaction. The method was developed during our efforts to synthesize a series of novel FKBP-12 inhibitors in which the known ketoamide linker was replaced with sulfamide.