34614-71-6Relevant academic research and scientific papers
PRODRUGS OF FUSED HETEROCYCLIC INHIBITORS OF D-AMINO ACID OXIDASE
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Page/Page column 101; 102, (2011/02/26)
The invention relates to prodrugs of fused heterocyclic inhibitors of D-amino oxidase (DAAO) and methods of treating diseases and conditions, wherein modulation of D-amino acid oxidase activity, D-serine levels, D-serine oxidative products and NMDA receptor activity in the nervous system of a mammalian subject is effective.
Improved synthesis of amino acid and dipeptide chloromethyl esters using bromochloromethane
Gomes, Paula,Santos, Maria Isabel,Trigo, Maria Joaquina,Castanheiro, Raquel,Moreira, Rui
, p. 1683 - 1693 (2007/10/03)
Peptide chloromethyl esters are important compounds in prodrug synthesis. A simple, mild and efficient method for the synthesis of chloromethyl esters of N-blocked amino acids and dipeptides using exclusively bromochloromethane is reported. These N-blocke
Chloromethyl ester of penicillins
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, (2008/06/13)
New penicillin esters and their salts together with methods for, and intermediates in the preparation thereof, the esters having the formula: EQU1 in which formula the asterisk indicates the possibility of an asymmetric carbon atom, n indicates an integer
