365545-15-9Relevant academic research and scientific papers
Aspartic protease inhibitors: Expedient synthesis of 2-substituted statines
Travins, Jeremy M.,Bursavich, Matthew G.,Veber, Daniel F.,Rich, Daniel H.
, p. 2725 - 2728 (2007/10/03)
(Equation presented) General stereocontrolled synthesis of all four (2,3)-stereoisomers of 2-substituted statines is described. The 2,3-syn and 2,3-anti isomers were synthesized via β-ketoester reduction and aldol reactions, respectively. Peptides contain
