3680-96-4Relevant articles and documents
A facile preparation of trisubstituted amino-furan and -thiophene derivatives
Medimagh, Raouf,Marque, Sylvain,Prim, Damien,Chatti, Saber
scheme or table, p. 6055 - 6065 (2011/10/08)
β-Alkylation of amino-furan and -thiophene heterocycles is described through metal-, acid- and base-free carbon-carbon bond formation. The ability of both heterocycles to undergo selective β-alkylation is compared by mean of experimental and theoretical data. The presence of chiral amine substituents induced the diastereoselective generation of the newly formed additional stereocenter.
BCRP/ABCG2 INHIBITOR
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Page/Page column 17, (2008/06/13)
The present invention is directed to a breast cancer resistance protein (BCRP/ABCG2) inhibitor. The BCRP inhibitor contains, as an active ingredient, an acrylonitrile derivative represented by formula (1): wherein one of R1 and R2 re
Ring-Chain Isomerism of N-(2-Hydroxyalkyl)nitrones, III. Nitrones of 2-Furancarbaldehydes
Kliegel, Wolfgang,Enders, Bernhard,Becker, Harald
, p. 27 - 45 (2007/10/02)
The ring-chain isomerism of N-(2-hydroxyalkyl)nitrones 3, obtained from 2-furancarbaldehyde and its 5-dialkylamino and 5-nitro derivatives, is studied by acylation of 3 with diphenylborinic acid, carboxylic acids, and isocyanates.Dependent on the kind of