391882-60-3Relevant academic research and scientific papers
Fancy bioisosteres: Metallocene-derived G-protein-coupled receptor ligands with subnanomolar binding affinity and novel selectivity profiles
Schlotter, Karin,Boeckler, Frank,Hübner, Harald,Gmeiner, Peter
, p. 3696 - 3699 (2005)
Metallocene-derived bioisosteres lead to exceptionally strong binding G-protein-coupled receptor ligands, indicating substantial plasticity of the receptor excluded volume. Novel binding profiles of ferrocenylcarboxamides combining subnanomolar Ki/s
A series of 18F-labelled pyridinylphenyl amides as subtype-selective radioligands for the dopamine D3 receptor
Hocke, Carsten,Maschauer, Simone,Huebner, Harald,Loeber, Stefan,Utz, Wolfgang,Kuwert, Torsten,Gmeiner, Peter,Prante, Olaf
scheme or table, p. 941 - 948 (2011/02/23)
Synthesis, biological activity, and structure-selectivity relationship (SSR) studies of a novel series of potential dopamine D3 receptor radioligands as imaging agents for positron emission tomography (PET) are reported. Considering a structurally diverse
INDOLIZINE CARBOXAMIDES AND THE AZA AND DIAZA DERIVATIVES THEREOF
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Page/Page column 56, (2010/10/19)
The invention relates to neuroreceptor-active carboxamide-substituted indolizine derivatives of general formula (I) wherein X represents a group of general formula (X1).
AZAINDOLE CARBOXAMIDES
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Page/Page column 33-35, (2010/11/30)
The invention relates to azaindole derivatives of general formula (I), wherein X represents a group of general formula (X1). Said compounds have a therapeutic potential in the treatment of diseases that are accompanied by an impaired dopamine metabolism a
