398145-88-5Relevant articles and documents
New serotonin 5-HT2A, 5-HT2B, and 5-HT2C receptor antagonists: Synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo and heterocycloalkanones
Brea,Rodrigo,Carrieri,Sanz,Cadavid,Enguix,Villazón,Mengod,Caro,Masaguer,Ravi?a,Centeno,Carotti,Loza
, p. 54 - 71 (2007/10/03)
A series of 52 conformationally constrained butyrophenones have been synthesized and pharmacologically tested as antagonists at 5-HT2A, 5-HT2B, and 5-HT2C serotonin receptors, useful for dissecting the role of each 5-HTsu