39887-56-4Relevant academic research and scientific papers
Synthesis and anion recognition studies of new oligomethylene bis(nitrophenylureylbenzamide) receptors
García-Elías, José,Ochoa-Terán, Adrián,Yatsimirsky, Anatoli K.,Santacruz Ortega, Hisila,Ochoa-Lara, Karen,López-Martínez, Luis Miguel,Castro-Riquelme, Christian L.,García, ángel L.,Madrigal-Peralta, Domingo,Labastida-Galván, Victoria,Ordo?ez, Mario
, p. 39147 - 39162 (2019/12/15)
A new series of oligomethylene bis(nitrophenylureylbenzamide) receptors were synthesized varying the relative position of the urea and amide groups (ortho4 and meta8) and the length of the oligomethylene chain (C2 to C8). An anion re
The parmodulin NRD-21 is an allosteric inhibitor of PAR1 Gq signaling with improved anti-inflammatory activity and stability
Gandhi, Disha M.,Rosas, Ricardo,Greve, Eric,Kentala, Kaitlin,D.-R. Diby, N'Guessan,Snyder, Vladyslava A.,Stephans, Allison,Yeung, Teresa H.W.,Subramaniam, Saravanan,DiMilo, Elliot,Kurtenbach, Khia E.,Arnold, Leggy A.,Weiler, Hartmut,Dockendorff
supporting information, p. 3788 - 3796 (2019/07/17)
Novel analogs of the allosteric, biased PAR1 ligand ML161 (parmodulin 2, PM2) were prepared in order to identify potential anti-thrombotic and anti-inflammatory compounds of the parmodulin class with improved properties. Investigations of structure-activi
Benzimidazolium-based receptors: Case of iodide-water cluster induced supramolecular chain and improved fluorometric binding of iodide involving alcoholic group
Ghosh, Kumaresh,Saha, Indrajit
, p. 57 - 65 (2013/06/26)
Benzimidazolium-based receptors 1 and 2 have been designed and synthesized. Anion binding studies reveal their selective fluorescence sensing of iodide in the excited state by exhibiting greater quenching of emission of anthracene. In the ground state, they prefer to bind bromide ion. Incorporation of alcoholic -OH in 2 leads to better performance over the receptor 1. The cyclooctameric structure as constituted by inclusion water and iodide interaction leads to ID-supramolecular chain with the structure 1 in the solid state. 1H NMR, UV-vis and fluorescence spectroscopic methods were adopted to study the anion binding behavior.
A new benzimidazolium receptor for fluorescence sensing of iodide
Ghosh, Kumaresh,Saha, Indrajit
scheme or table, p. 311 - 317 (2010/10/18)
A new anthracene-appended benzimidazolium-based receptor 1 has been designed and synthesised. The receptor shows selective recognition of iodide in the excited state by exhibiting quenching of emission of anthracene. In the ground state, receptor 1 shows
A mild and clean method for oxidative formation of amides from aldehydes and amines
Fang, Chen,Qian, Weixing,Bao, Weiliang
experimental part, p. 2529 - 2531 (2009/04/12)
A metal-free direct oxidative formation of amides from aldehydes and amines using a hypervalent iodine(III) reagent or an ion-supported hypervalent iodine(III) reagent as a recyclable oxidant under mild conditions is reported. Georg Thieme Verlag Stuttgart.
3-(2′-Bromopropionylamino)-benzamides as novel S-phase arrest agents
Hu, Laixing,Li, Zhuo-rong,Li, Jian-Nong,Qu, Jinrong,Jiang, Jian-Dong,Boykin, David W.
, p. 6847 - 6852 (2008/09/16)
We report the synthesis, antiproliferative activity, and SAR of novel 3-(2′-bromopropionylamino)-benzamides. Many of the benzamide compounds showed potent cytotoxicities against Molt-3 leukemia cells. Several compounds exihibited cytotoxicities (under 6.5
Thermosensitive recording material and novel color developer compounds
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, (2008/06/13)
Disclosed is a thermosensitive recording material comprising a sheet-shaped support and a thermosensitive recording layer which is formed on at least one surface of the support and comprises a colorless or light-colored dye precursor and a color developer capable of reacting with the dye precursor and inducing color formation therein upon application of heat thereto, the color developer comprising a compound represented by the following formula (I) or analog thereof:: The thermosensitive recording material has high sensitivity and can prevent white background portions from coloring and recorded images from decolorizing in an environmental resistance test.
11a-Methano-TXA compounds
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, (2008/06/13)
The present invention provides novel 11a-methano-TXA compounds and intermediates and processs for their preparation. Further provided are methods for using these novel TXA analogs as inhibitors of thromboxane synthetase, rendering these analogs useful for a variety of pharmacological purposes. These pharmacological uses include anti-inflammatory, anti-thromobitc, and anti-asthma indications.
