405872-78-8 Usage
Uses
Used in Pharmaceutical Applications:
Ethyl 2-chloro-2-(2-(3-methoxyphenyl)hydrazono)acetate is used as a potent and selective ligand for the δ opioid receptor. This application is significant because the δ opioid receptor plays a crucial role in various physiological processes and has been implicated in pain management, addiction, and other neurological disorders. By acting as a selective ligand, ethyl 2-chloro-2-(2-(3-methoxyphenyl)hydrazono)acetate can potentially be used to modulate the activity of the δ opioid receptor, offering new therapeutic strategies for treating related conditions.
Used in Research and Development:
In addition to its potential pharmaceutical applications, ethyl 2-chloro-2-(2-(3-methoxyphenyl)hydrazono)acetate can also be used as a research tool to better understand the structure and function of the δ opioid receptor. ethyl 2-chloro-2-(2-(3-methoxyphenyl)hydrazono)acetate can be employed in various experimental setups, such as binding assays, functional assays, and cell-based assays, to investigate the receptor's properties and its interactions with other molecules. This knowledge can contribute to the development of more effective and targeted therapies for conditions related to the δ opioid receptor.
Used in Drug Design and Optimization:
The unique chemical structure of ethyl 2-chloro-2-(2-(3-methoxyphenyl)hydrazono)acetate makes it a valuable starting point for the design and optimization of new drugs targeting the δ opioid receptor. By exploring the structure-activity relationships of ethyl 2-chloro-2-(2-(3-methoxyphenyl)hydrazono)acetate, researchers can identify key structural features that contribute to its potency and selectivity. This information can then be used to guide the design of more effective and safer drugs with improved pharmacological properties.
Check Digit Verification of cas no
The CAS Registry Mumber 405872-78-8 includes 9 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 6 digits, 4,0,5,8,7 and 2 respectively; the second part has 2 digits, 7 and 8 respectively.
Calculate Digit Verification of CAS Registry Number 405872-78:
(8*4)+(7*0)+(6*5)+(5*8)+(4*7)+(3*2)+(2*7)+(1*8)=158
158 % 10 = 8
So 405872-78-8 is a valid CAS Registry Number.
405872-78-8Relevant academic research and scientific papers
Novel delta opioid receptor agonists exhibit differential stimulation of signaling pathways
Peng, Youyi,Zhang, Qiang,Arora, Sonia,Keenan, Susan M.,Kortagere, Sandhya,Wannemacher, Kenneth M.,Howells, Richard D.,Welsh, William J.
experimental part, p. 6442 - 6450 (2011/02/26)
A novel family of 1,3,5-trisubstituted 1,2,4-triazoles was discovered as potent and selective ligands for the δ opioid receptor by rational design. Compound 5b exhibited low-nanomolar in vitro binding affinity (IC50 = 5.8 nM), excellent selecti
OPIOID RECEPTOR SUBTYPE-SELECTIVE AGENTS
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Page/Page column 34, (2008/06/13)
Opioid receptor compounds and pharmaceutical compositions thereof are presented. Also presented are methods for treating a condition mediated by an opioid receptor by administering an effective amount of the opioid receptor compound to a patient in need thereof.
