41339-64-4Relevant articles and documents
E-SELECTIN ANTAGONISTS
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Page/Page column 47, (2012/04/04)
Compounds, compositions and methods are provided for inhibiting in vitro and in vivo processes mediated by E-selectin binding. More specifically, particular glycomimetic compounds are described, wherein the compounds are E- selectin antagonists.
First heterogeneous ligand- and salt-free larock indole Synthesis
Batail, Nelly,Bendjeriou, Anissa,Lomberget, Thierry,Barrett, Roland,Dufaud, Veronique,Djakovitch, Laurent
supporting information; experimental part, p. 2055 - 2062 (2009/12/26)
A new ligand- and salt-free procedure using heterogeneous palladium catalysts for the Larock indole and benzofuran synthesis is reported. After optimisation of the reaction conditions, good to high isolated yields have been achieved for a variety of structures. Recycling studies have shown that the palladium catalysts can be readily recovered and reused. Reactions and recovery of the palladium catalysts can be carried out in the presence of air, without any particular precaution.
Indolylalkylpiperidines
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, (2008/06/13)
1-(Indolyl-3-alkyl)-3 or 4-(ureido or guanidino)-piperidines, e.g. those of the formula STR1 R= H; alkyl; free, etherified or esterified OH or SH; CF3, NO2 or NH2 m= 1-4; n= 2 or 3; X= O, S or NH acyl derivatives and salts thereof are antihypertensive agents.