419555-07-0Relevant academic research and scientific papers
Intramolecular olefin diamination for the stereoselective synthesis of 3-aminopiperidines
Kong, Aidi,Blakey, Simon B.
experimental part, p. 1190 - 1198 (2012/05/20)
A general method for the direct intramolecular diamination of terminal olefins is presented. The reaction, mediated by hypervalent iodine oxidants, produces substituted 3-aminopiperidine scaffolds with high regio- and stereoselectivity, rendering this process relevant to both medicinal chemistry and natural products synthesis. Georg Thieme Verlag Stuttgart New York.
