428478-01-7Relevant academic research and scientific papers
Enantioselective N-Acylation of Biginelli Dihydropyrimidines by Oxidative NHC Catalysis
Brandolese, Arianna,Ragno, Daniele,Leonardi, Costanza,Di Carmine, Graziano,Bortolini, Olga,De Risi, Carmela,Massi, Alessandro
, p. 2439 - 2447 (2020)
The oxidative N-acylation reaction of 3,4-dihydropyrimidin-2-(1H)-ones (DHPMs) with enals and N-heterocyclic carbene (NHC) catalysts is described. The reaction proceeds in the presence of quinone oxidant without additional acyl transfer agents and in the
