496064-28-9Relevant articles and documents
Synthesis and biological evaluation of anthranilamide-based non-peptide mimetics of ω-conotoxin GVIA
Baell, Jonathan B.,Duggan, Peter J.,Forsyth, Stewart A.,Lewis, Richard J.,Lok, Y. Phei,Schroeder, Christina I.,Shepherd, Nicholas E.
, p. 7284 - 7292 (2007/10/03)
Non-peptide mimetics based on an anthranilamide 'scaffold' possessing fragments that mimic Lys2, Tyr13 and Arg17 in ω-conotoxin GVIA have been prepared. Compounds were assayed for binding to the voltage-gated calcium channels Cav2.2 ('N-type')