503186-56-9Relevant academic research and scientific papers
2,6-Dimethyltyrosine analogues of a stereodiversified ligand library: Highly potent, selective, non-peptidic μ opioid receptor agonists
Harrison, Bryce A.,Pasternak, Gavril W.,Verdine, Gregory L.
, p. 677 - 680 (2003)
We recently reported the use of an exhaustively stereodiversified library based on endomorphin-2 (1) to discover μ opioid receptor (MOR) ligands of type 2-4. Here, we report the synthesis and evaluation of 2,6-dimethyltyrosine analogues 5-10. These analog
MU OPIOID RECEPTOR LIGANDS: METHODS OF USE AND SYNTHESIS
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Page 68-70, (2008/06/13)
Peptidomimetic compounds derived from aralkyl substitued 8-amino-3,7- or 3,6-dihydroxy alkenoic or alkanoic acids and compositions including those compounds, as well as methods of using and making the compounds are herein described. The compounds are usef
