512773-83-0Relevant articles and documents
Nucleophilic substitution reaction in indole chemistry: 1-methoxy-6-nitroindole-3-carbaldehyde as a versatile building block for 2,3,6-trisubstituted indoles
Yamada, Koji,Yamada, Fumio,Shiraishi, Takei,Tomioka, Saori,Somei, Masanori
experimental part, p. 971 - 982 (2010/10/03)
1-Methoxy-6-nitroindole-3-carbaldehyde is proved to be a versatile electrophile and reacts regioselectively at the 2-position with various types of nucleophiles providing 2,3,6-trisubstituted indole derivatives. The reaction is applicable for the preparation of a novel pyrimido[1,2-a]indole derivative.