5584-30-5Relevant academic research and scientific papers
Studies with enamines: Route to aminoazolopyrimidines and arylazoazolopyrimidines
Salaheldin, Abdellatif M.,Khairou, Khalid S.
, p. 175 - 181 (2013/04/23)
An easy preparation of enaminonitrile derivatives and their transformation into new substituted azolopyrimidines is described. The one-step transformation was carried out under microwave irradiation and by classical heating methods. The use of microwave i
Enaminonitriles in heterocyclic synthesis: A route to 1,3-diaryl-4- Aminopyrazole derivatives
Medrasi, Hanadi Y.,Al-Sheikh, Mariam Abdullah,Salaheldin, Abdellatif Mohamed
, p. 535 - 544 (2013/03/13)
Benzylcyanide and 4-nitrobenzylcyanide condensed with triethyl orthoformate and piperidine or morpholine to yield 2-Aryl-2-piperidinyl or 2-morpholinylacrylonitriles. These coupled with aromatic diazonium salts to yield the 2-Arylhydrazno-2-Arylethane nit
New pyrazolo[1,5a]pyrimidines as orally active inhibitors of Lck
Gommermann, Nina,Buehlmayer, Peter,Von Matt, Anette,Breitenstein, Werner,Masuya, Keiichi,Pirard, Bernard,Furet, Pascal,Cowan-Jacob, Sandra W.,Weckbecker, Gisbert
scheme or table, p. 3628 - 3631 (2010/09/04)
A novel series of pyrazolo[1,5a]pyrimidines was optimized to target lymphocyte-specific kinase (Lck). An efficient synthetic route was developed and SAR studies toward activity and selectivity are described, leading to Lck inhibitors with enzymatic, cellu
7-Aminopyrazolo[1,5-a]pyrimidines as potent multitargeted receptor tyrosine kinase inhibitors
Frey, Robin R.,Curtin, Michael L.,Albert, Daniel H.,Glaser, Keith B.,Pease, Lori J.,Soni, Niru B.,Bouska, Jennifer J.,Reuter, David,Stewart, Kent D.,Marcotte, Patrick,Bukofzer, Gail,Li, Junling,Davidsen, Steven K.,Michaelides, Michael R.
experimental part, p. 3777 - 3787 (2009/04/07)
7-Aminopyrazolo[1,5-a]pyrimidine urea receptor tyrosine kinase inhibitors have been discovered. Investigation of structure-activity relationships of the pyrazolo[1,5-a]pyrimidine nucleus led to a series of 6-(4-N,N′-diphenyl) ureas that potently inhibited
PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES AND THEIR THERAPEUTIC USE
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Page/Page column 8, (2008/06/13)
Disclosed are pyrazolo-pyrimidine derivatives which have interesting pharmaceutical properties.
