56877-16-8

Upstream product

• 56877-15-7 (1,3-Dimethyl-5-methylamino-1H-pyrazol-4-yl)-(2-fluoro-phenyl)-methanone 
• 598-21-0 2-Bromoacetyl bromide 

Downstream Products

• 103068-95-7 4-(2-Fluoro-phenyl)-1,3,7-trimethyl-5-[3-(2-methyl-piperidin-1-yl)-propylamino]-1,7-dihydro-pyrazolo[3,4-b]pyridin-6-one 
• 103068-89-9 N-[4-(2-Fluoro-benzoyl)-2,5-dimethyl-2H-pyrazol-3-yl]-N-methyl-2-[3-(2-methyl-piperidin-1-yl)-propylamino]-acetamide 

Relevant academic research and scientific papers

Pyrazolodiazepines. 2. 4-Aryl-1,3-dialkyl-6,8-dihydropyrazolo[3,4-e][1,4]diazepin-7(1H)-ones as antianxiety and anticonvulsant agents

A series of 4-aryl-1,3-dialkyl-6,8-dihydropyrazolo[3,4-e][1,4] diazepin-7(1H)-ones was synthesized and screened for psychotropic activity. In animals, a number of these pyrazolodiazepinones had strong CNS effects similar to diazepam. One compound, 4-(2-fluorophenyl)-6,8-dihydro-1,3,8 trimethylpyrazolo[3,4-e][1,4)diazepin-7(1H)-one (54), is being studied in the clinic as a component of a new animal anesthetic Tilazol.