57036-35-8Relevant academic research and scientific papers
Synthesis of novel GABA uptake inhibitors. 3. Diaryloxime and diarylvinyl ether derivatives of nipecotic acid and guvacine as anticonvulsant agents
Knutsen, Lars J. S.,Andersen, Knud Erik,Lau, Jesper,Lundt, Behrend F.,Henry, Rodger F.,Morton, Howard E.,N?rum, Lars,Petersen, Hans,Stephensen, Henrik,Suzdak, Peter D.,Swedberg, Michael D. B.,Thomsen, Christian,S?rensen, Per O.
, p. 3447 - 3462 (2007/10/03)
(3R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid 1 (tiagabine, Gabitril) is a potent and selective γ-aminobutyric acid (GABA) uptake inhibitor with proven anticonvulsant efficacy in humans. This drug, which has a unique mechanism
Amino acid derivatives
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, (2008/06/13)
Compounds of the Formula I STR1 wherein R1 represents phenyl, or phenyl substituted by one, or more substituents selected from the group consisting of halogen, C1-7 -alkyl, and C1-7 -alkoxy, R2 represents furany
