573716-83-3

Upstream product

• 205813-79-2 tert-butyl (3aR,4S,7R,7aS)-2,2-dimethyl-5-[(4-methylphenyl)sulfonyl]-3a,4,7,7a-tetrahydro-4,7-epimino-1,3-benzodioxole-8-carboxylate 
• 573716-76-4 (-)-(1S,2R,3S,4R,5S,6R)-7-tert-butoxycarbonyl-2,3-exo-isopropylidenedioxy-5-endo-methanesulfonyloxy-6-endo-p-toluenesulfonyl-7-azabicyclo[2.2.1]heptane 
• 573716-64-0 tert-butyl (1S,2R,3S,4R,5S,6R)-2,3,5-trihydroxy-6-[(4-methylphenyl)sulfonyl]-7-azabicyclo[2.2.1]heptane-7-carboxylate 
• 573717-23-4 tert-butyl (1R,4S,5R,6S)-5-[(4-methylphenyl)sulfonyl]-6-({[(1S,4R)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]hept-1-yl]carbonyl}oxy)-7-azabicyclo[2.2.1]hept-2-ene-7-carboxylate 
• 573716-70-8 (-)-(1S,2R,3S,4R,5S,6R)-7-tert-butoxycarbonyl-2,3-exo-isopropylidenedioxy-6-endo-p-toluenesulfonyl-7-azabicyclo[2.2.1]heptane-5-endo-ol 
• 573716-62-8 tert-butyl (1S,4R,5S,6R)-5-hydroxy-6-[(4-methylphenyl)sulfonyl]-7-azabicyclo[2.2.1]hept-2-ene-7-carboxylate 
• 227454-54-8 5-oxo-6-(toluene-4-sulfonyl)-7-aza-bicyclo[2.2.1]hept-2-ene-7-carboxylic acid tert-butyl ester 

Downstream Products

• 599199-70-9 (1R,2R,6S,7R)-4,4-Dimethyl-3,5-dioxa-8,11-diaza-tricyclo[5.3.1.0^2,6]undec-8-ene-11-carboxylic acid tert-butyl ester 
• 599199-71-0 (1R,2R,6S,7R)-4,4-Dimethyl-3,5-dioxa-8,11-diaza-tricyclo[5.3.1.0^2,6]undecane-11-carboxylic acid tert-butyl ester 
• 599199-75-4 (1S,2R,6S,7S,8R,9S)-8-Amino-4,4-dimethyl-9-(toluene-4-sulfonyl)-3,5-dioxa-10-aza-tricyclo[5.2.1.0^2,6]decane-10-carboxylic acid tert-butyl ester 

Relevant academic research and scientific papers

Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues

Enantiomerically pure alcohols (-)- and (+)-7-tert-butoxycarbonyl-6-endo-p-toluenesulfonyl-7-azabicyclo[2.2.1] hept-2-en-5-endo-ol ((-)-11 and (+)-11) have been obtained from the Diels-Alder adduct of N-(tert-butoxycarbonyl)pyrroel and 2-bromo-1-p-toluene