579525-46-5Relevant articles and documents
Facile Palladium-Catalyzed Synthesis of 3-Arylpyrazolo-[1,5-a]pyrimidines
Majo, Vattoly J.,Prabhakaran, Jaya,John Mann,Dileep Kumar
, p. 620 - 624 (2003)
An efficient palladium-catalyzed synthesis of 3-arylpyrazolo[1,5-a] pyrimidines has been investigated. The key step in the synthesis is a Suzuki biaryl coupling of 3-bromo-2,5-dimethyl-7-aminopyrazolo[1,5-a]pyrimidines with arylboronic acids to provide 3-
ANTI-MALIGNANT TUMOR AGENT COMPOSITION
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Paragraph 0087; 0109, (2016/01/25)
To provide a satisfactory anticancer agent composition suppressing the growth of cancer (malignant tumor) reliably and hardly causing side effects, the present invention is directed to an anticancer agent composition including the following agents as active ingredient; a LAT1 inhibitor, and one or more agents selected from the group consisting of an alkylating agent, a platinum-based antineoplastic agent, an anti-metabolite, a topoisomerase inhibitor, an anti-microtubule polymerizing agent, a hormonal agent, an anti-microtubule depolymerizing agent, an anticancer antibiotic, and a molecular targeted agent.
SUBSTITUTED PYRIDOPYRAZINES AS NOVEL SYK INHIBITORS
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Page/Page column 36, (2013/02/27)
Provided are certain pyridopyrazine compounds, pharmaceutical compositions thereof and methods of use therefor.