59440-79-8Relevant articles and documents
Potent hFPRL1 (ALXR) agonists as potential anti-inflammatory agents
Buerli, Roland W.,Xu, Han,Zou, Xiaoming,Muller, Kristine,Golden, Jennifer,Frohn, Mike,Adlam, Matthew,Plant, Matthew H.,Wong, Min,McElvain, Michele,Regal, Kelly,Viswanadhan, Vellarkad N.,Tagari, Philip,Hungate, Randall
, p. 3713 - 3718 (2007/10/03)
We report the discovery of potent agonists for the human formyl-peptide-like 1 receptor (hFPRL1). These compounds did not act at a closely related receptor denoted human formyl peptide receptor (hFPR) up to 10 μM concentration. Recent studies have indicat
NOVEL UREIDO - AND AMIDO-PYRAZOLONE DERIVATIVES
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Page 24-25, (2008/06/13)
The present invention provides compounds of formula (I); wherein each of R1 to R4 is independently selected from hydrogen, a halogen, a substituted or unsubstituted cyclic and heterocyclic moiety, substituted or unsubstituted, linear or branched alkyl, alkyloxy, alkylcarbonyl, alkyloxycarbonyl, alkenyl, alkenyloxy, alkenylcarbonyl, alkenyloxycarbonyl, alkynyl, alkynyloxy, alkynylcarbonyl, alkynyloxycarbonyl, aryl, benzyl, arlyoxy, arylcarbonyl, aryloxycarbonyl and sulphur equivalents of said oxy, carbonyl and oxycarbonyl moieties, and A is NH, or (CH2)n, where n is preferably 0, 1 or 2. The invention also relates to methods for preparing the compounds and their uses as CCK receptor ligands and CCK antagonists.