616898-54-5

Basic information

• Product Name: no
• Synonyms: C8813;Cyclohexanol, 4-(4-broMophenyl)-4-(diMethylaMino)-1-[2-(2-thienyl)ethyl]-, trans-;(1r,4r)-4-(4-bromophenyl)-4-(dimethylamino)-1-(2-(thiophen-2-yl)ethyl)cyclohexanol
• CAS NO: 616898-54-5
• Molecular Formula: C20H26BrNOS
• Molecular Weight: 408.39554
• Product Categories: Amines;Aromatics;Intermediates & Fine Chemicals;Neurochemicals;Pharmaceuticals
• Mol File: 616898-54-5.mol
• Article Data: 0

Chemical Properties

• Appearance: /
• Storage Temp.: Refrigerator
• Solubility: Chloroform, Methanol
• CAS DataBase Reference: no(CAS DataBase Reference)
• NIST Chemistry Reference: no(616898-54-5)
• EPA Substance Registry System: no(616898-54-5)

Safety Data

• Hazardous Substances Data: 616898-54-5(Hazardous Substances Data)

Usage

Description

Thiobromadol is a synthetic opioid analgesic that is a derivative of the opioid drug Bromptramol. It is designed to provide potent pain relief while minimizing the risk of addiction and abuse. Thiobromadol is a high affinity agonist for the μand δ-opioid receptors, but has almost no affinity for the κ-opioid receptor.

Uses

Used in Pain Management:
Thiobromadol is used as a potent analgesic for the management of moderate to severe pain. Its high affinity for the μand δ-opioid receptors allows it to effectively alleviate pain while reducing the risk of addiction and abuse compared to traditional opioids.
Used in Pharmaceutical Industry:
Thiobromadol is used in the development of new pharmaceutical drugs for pain management. Its unique properties and reduced potential for abuse make it a promising candidate for the creation of safer and more effective pain relief medications.
Used in Research:
Thiobromadol is also used in scientific research to study the mechanisms of opioid analgesia and addiction. Its selective action on the μand δ-opioid receptors provides valuable insights into the development of new drugs with improved safety profiles and reduced potential for abuse.