623950-07-2Relevant articles and documents
Identification of potent phenyl imidazoles as opioid receptor agonists
Breslin, Henry J.,Cai, Chaozhong,Miskowski, Tamara A.,Coutinho, Santosh V.,Zhang, Sui-Po,Hornby, Pamela,He, Wei
, p. 2505 - 2508 (2006)
Using previously reported opioid receptor (OR) agonist analogs 4a-c as starting points, the structure-activity relationship (SAR) for their related series has been further refined. This SAR study has led to the identification of 2,6-di-Me-Tyr (DMT) analog
Novel compounds as opioid receptor modulators
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Page/Page column 33, (2010/02/05)
This invention is directed towards novel compounds as opioid receptor modulators, antagonists, and agonists useful for the treatment of opioid modulated disorders such as pain and gastrointestinal disorders.