6243-59-0Relevant academic research and scientific papers
ARYL HYDROCARBON RECEPTOR MODULATORS AND USES THEREOF
-
Paragraph 00426; 00450, (2019/10/29)
Provided are compounds of Formula (I), and pharmaceutically acceptable salts, solvates, hydrates, stereoisomers, tautomers, isotopically labeled derivatives, polymorphs, and prodrugs thereof, wherein X1-X4, RX, RC, RB, n, and Ring A are as defined herein. The compounds may be aryl hydrocarbon receptor agonists or partial aryl hydrocarbon receptor agonists. Also provided are pharmaceutical compositions comprising a compound of Formula (I) and methods of using such compounds for treating diseases and conditions related to the activity of an aryl hydrocarbon receptor, such as, for example, inflammatory diseases, autoimmune diseases, metabolic disorders, and proliferative diseases.
A Novel Total Synthesis of Indolo[2,3-b]naphthalene-6,11-diones
Fernandez, Marcos,Barcia, Carlos,Estévez, Juan C.,Estévez, Ramón J.,Castedo, Luis
, p. 267 - 270 (2007/10/03)
A new total synthesis of indolo[2,3-b]naphthalene-6,11-diones is described, which involves a novel opening of 2-(2′-nitrophenyl)-2-methoxycarbonyl-1- indanones to 2-[2-memoxycarbonyl-2-(2-nitrophenyl)ethyl]benzoic acids followed by a two-steps transformat
Synthesis, electrochemistry, and bioactivity of the cyanobacterial calothrixins and related quinones
Bernardo, Paul H.,Chai, Christina L. L.,Heath, Graham A.,Mahon, Peter J.,Smith, Geoffrey D.,Waring, Paul,Wilkes, Bronwyn A.
, p. 4958 - 4963 (2007/10/03)
The calothrixins are quinone-based natural products isolated from Calothrix cyanobacteria which show potent antiproliferative properties against several cancer cell lines. Preliminary mechanistic studies suggest that the biological mode of action of the c
