644988-83-0Relevant articles and documents
Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype
Hocke, Carsten,Prante, Olaf,Loeber, Stefan,Huebner, Harald,Gmeiner, Peter,Kuwert, Torsten
, p. 3963 - 3966 (2007/10/03)
Starting from FAUC 365, a series of iodine substituted heteroaryl carboxamides has been synthesized revealing high affinity and selectivity for the dopamine D3 receptor. Binding data showed a 15-560-fold selectivity for the dopamine D3 over D2. A 2,3-dich