65133-71-3Relevant academic research and scientific papers
Synthesis of 4-Acyl-2,3-dihydro-4H-1,4-oxazines
Nicola, Massimo,Gaviraghi, Giovanni,Pinza, Mario,Pifferi, Giorgio
, p. 825 - 828 (2007/10/02)
The synthesis of 4-acyl-2,3-dihydro-4H-1,4-oxazines (6a-h) via acid dehydration of 4-acyl 2- and 3-morpholinols is described.During dehydration of 2-morpholinols 3d,e, N-alkylisoquinolones 7a-e were also isolated.
Synthesis of N-alkoxybenzoylmorpholinols as possible metabolites of trithiozine.
Gaviraghi,Nicola,Pinza,Pifferi
, p. 801 - 811 (2007/10/02)
The synthesis of some possible metabolites of trithiozine, a new antisecretory-antiulcer drug, is reported. The metabolite 4-(3,4,5-trimethoxybenzoyl)-2-morpholinol (III a) was prepared by oxidative cyclization of the corresponding diethanolamine derivati
