65376-39-8Relevant academic research and scientific papers
Synthesis of some amino acid and peptide conjugates and their evaluation as potential anti-allergic and anti-inflammatory agents
Shalaby,Abd Al-Salam,Kalmouch,El-Shihaby,Abdullah
, p. 401 - 415 (2015/10/20)
ANEW series of N-3-(2-furanyl) acryloyl, N-3-(5-methyl)-2-(furanyl)-acryoyl amino acids, peptide and piprazines amids, were structurally designed and synthesized. About 23 compounds (5a-w) were synthesized and their anti-allergic and anti-inflamatory acti
Carboxamidation of carboxylic acids with 1-tert-butoxy-2-tert-butoxycarbonyl-1,2-dihydroisoquinoline (BBDI) without bases
Saito, Yukako,Ouchi, Hidekazu,Takahata, Hiroki
experimental part, p. 11129 - 11135 (2009/04/11)
Formation of carboxamides of a variety of carboxylic acids with the coupling reagent BBDI is described. This procedure permits a one pot and simple operation without the need of any bases and no base was?required for even use of amine hydrochlorides. In addition, an approach to BBDI-catalyzed carboxamidation is examined.
