65687-00-5 Usage
Description
(-)-4,5-dihydro-N-(2,2,2-trifluoro-1-phenylethyl)oxazol-2-amine, also known as tapentadol, is a synthetic opioid analgesic that possesses both mu-opioid receptor agonist and norepinephrine reuptake inhibitor activity. This dual mechanism of action allows it to provide both opioid and non-opioid analgesia, making it a versatile pain management option.
Uses
Used in Pain Management:
Tapentadol is used as an analgesic agent for the treatment of moderate to severe acute pain and chronic pain conditions, such as neuropathic pain and musculoskeletal pain. Its unique dual mechanism of action allows for effective pain relief by targeting both opioid receptors and inhibiting the reuptake of norepinephrine, leading to enhanced analgesic effects.
Used in Pharmaceutical Industry:
In the pharmaceutical industry, tapentadol is utilized as an active pharmaceutical ingredient in the development of pain management medications. It is available in various forms, including immediate-release and extended-release tablets, to cater to different patient needs and ensure optimal dosing regimens.
Used in Controlled Substances:
Due to its potential for abuse and addiction, tapentadol is considered a controlled substance. As such, it is typically prescribed under the supervision of a healthcare professional to ensure safe and effective use while minimizing the risk of misuse and dependence.
Check Digit Verification of cas no
The CAS Registry Mumber 65687-00-5 includes 8 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 5 digits, 6,5,6,8 and 7 respectively; the second part has 2 digits, 0 and 0 respectively.
Calculate Digit Verification of CAS Registry Number 65687-00:
(7*6)+(6*5)+(5*6)+(4*8)+(3*7)+(2*0)+(1*0)=155
155 % 10 = 5
So 65687-00-5 is a valid CAS Registry Number.
InChI:InChI=1/C11H11F3N2O/c12-11(13,14)9(8-4-2-1-3-5-8)16-10-15-6-7-17-10/h1-5,9H,6-7H2,(H,15,16)
65687-00-5Relevant articles and documents
Aryltrifluoroethylamines
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, (2008/06/13)
Certain arylmethyl amines have been prepared wherein the "methyl" carbon is substituted with a polyfluoroalkyl radical. The compounds form acid addition salts, exist in resolvable stereoisomeric forms, and are useful for treating hypertension. Formulations for human and veterinary medicine are described, as well as methods of use.
