67752-29-8Relevant academic research and scientific papers
Plasmodium falciparum subtilisin-like protease 1: Discovery of potent difluorostatone-based inhibitors
Giovani, Simone,Penzo, Maria,Butini, Stefania,Brindisi, Margherita,Gemma, Sandra,Novellino, Ettore,Campiani, Giuseppe,Blackman, Michael J.,Brogi, Simone
, p. 22431 - 22448 (2015/06/02)
Currently available drugs to treat malaria are often ineffective due to the acquisition of drug resistance. In this context, drugs with innovative modes of action and no liability to cross-resistance are urgently needed. Recently, subtilisin-like protease
9A-SUBSTITUTED AZALIDES
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, (2008/06/13)
The present invention relates to novel 9a-substituted azalides having antimalarial activity. More particularly, the invention relates to 9a-substituted 9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A, 3-O-decladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythr
